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RECRUITING
NCT04104776
PHASE1/PHASE2

A Study of Tulmimetostat DZR123 (CPI-0209) in Patients With Advanced Solid Tumors and Lymphomas

Sponsor: Novartis Pharmaceuticals

View on ClinicalTrials.gov

Summary

The purpose of this open-label, first-in-human (FIH) trial is to evaluate the safety, tolerability, pharmacokinetics, pharmacodynamics, and preliminary antitumor activity of DZR123 (Tulmimetostat, CPI-0209), both as monotherapy and in combination with enzalutamide, in patients with advanced solid tumors and lymphomas.

Official title: A Phase 1/2 Study of DZR123 (CPI-0209) in Patients With Advanced Solid Tumors and Lymphomas

Key Details

Gender

All

Age Range

18 Years - Any

Study Type

INTERVENTIONAL

Enrollment

300

Start Date

2019-09-18

Completion Date

2030-02-27

Last Updated

2026-08-19

Healthy Volunteers

No

Interventions

DRUG

Tulmimetostat

Tulmimetostat dosed once per day orally in 28 day cycles

DRUG

Enzalutamide

Enzalutamide dosed once per day orally in 28 day cycles

Locations (80)

H. Lee Moffitt Cancer Center & Research Institute

Tampa, Florida, United States

Winship Cancer Institute of Emory University

Atlanta, Georgia, United States

University of Chicago Medical Center

Chicago, Illinois, United States

Loyola University Medical Center

Maywood, Illinois, United States

University of Maryland Greenebaum Cancer Center

Baltimore, Maryland, United States

Massachusetts General Hospital

Boston, Massachusetts, United States

Dana Farber Cancer Institute

Boston, Massachusetts, United States

University of Michigan Hospitals

Ann Arbor, Michigan, United States

South Texas Accelerated Research Therapeutics (START) - Midwest Location

Grand Rapids, Michigan, United States

Hackensack University Medical Center

Hackensack, New Jersey, United States

Roswell Park Cancer Institute

Buffalo, New York, United States

Laura and Isaac Perlmutter Cancer Center at NYU Langone

New York, New York, United States

Memorial Sloan Kettering Cancer Center - NYC

New York, New York, United States

Weill Medical College of Cornell University

New York, New York, United States

University of Rochester Medical Center, James P. Wilmot Cancer Center

Rochester, New York, United States

Montefiore Medical Center, Montefiore Medical Center Laboratories

The Bronx, New York, United States

University of Cincinnati Medical Center

Cincinnati, Ohio, United States

Abramson Cancer Center of the University of Pennsylvania

Philadelphia, Pennsylvania, United States

South Texas Accelerated Research Therapeutics

San Antonio, Texas, United States

University of Virginia Health System

Charlottesville, Virginia, United States

Swedish Cancer Institute

Seattle, Washington, United States

Fred Hutchinson Cancer Center

Seattle, Washington, United States

CHU Bordeaux Hopital Saint Andre

Bordeaux, France

CLCC Institut Bergonie

Bordeaux, France

Centre Oscar Lambret

Lille, France

Centre Leon Berard

Lyon, France

CHU Nantes Hopital Hotel Dieu

Nantes, France

CHU Nantes Hopital Nord Laennec

Saint-Herblain, France

Hopital Hautepierre

Strasbourg, France

Gustave Roussy

Villejuif, France

Irccs University Hospital of Bologna

Bologna, Italy

National Cancer Institute, IRCCS

Milan, Italy

National Cancer Institute, IRCCS

Milan, Italy

European Institute of Oncology (IEO), IRCCS

Milan, Italy

European Institute of Oncology (IEO), IRCCS

Milan, Italy

Humanitas San Pio X

Milan, Italy

University Polyclinic Foundation "Agostino Gemelli" - IRCCS

Roma, Italy

Gruppo Humanitas - Humanitas Research Hospital - Cancer Center

Rozzano, Italy

University Teaching Centre, Early Clinical Trials Unit

Gdansk, Poland

Pratia MCM Krakow

Krakow, Poland

Polish Mother's Memorial Hospital-Research Institute

Lodz, Poland

Pratia - Poznan

Poznan, Poland

University Teaching Hospital in Poznan, Department of Gynecologic Oncology

Poznan, Poland

Maria Sklodowska-Curie - National Research Institute of Oncology

Warsaw, Poland

Keimyung University - Dongsan Medical Center

Daegu, South Korea

National Cancer Center

Goyang-si, South Korea

Gachon University Gil Medical Center

Incheon, South Korea

Seoul National University Hospital

Seoul, South Korea

Severance Hospital, Yonsei University Health System

Seoul, South Korea

Asan Medical Center

Seoul, South Korea

Gangnam Severance Hospital

Seoul, South Korea

The Catholic University of Korea, Seoul St. Mary's Hospital

Seoul, South Korea

University Hospital Vall d'Hebron

Barcelona, Spain

Hospital Clinic of Barcelona

Barcelona, Spain

University Hospital of Girona Dr. Josep Trueta

Girona, Spain

Catalan Institute of Oncology, Hospital Duran i Reynals

L'Hospitalet de Llobregat, Spain

University Clinic of Navarra - Madrid

Madrid, Spain

University Hospital Ramon y Cajal

Madrid, Spain

University Hospital Clinical San Carlos, Department of Medical Oncology

Madrid, Spain

University Hospital Foundation Jimenez Diaz

Madrid, Spain

University Hospital 12 de Octubre

Madrid, Spain

University Hospital Quiron Madrid

Madrid, Spain

University Hospital Puerta de Hierro Majadahonda

Majadahonda, Spain

University Hospital Son Espases

Palma, Spain

University Clinic of Navarra - Pamplona

Pamplona, Spain

Parc Tauli Health Corporation

Sabadell, Spain

University Clinical Hospital of Salamanca

Salamanca, Spain

University Hospital Complex of Santiago (CHUS)

Santiago de Compostela, Spain

University Hospital Virgen del Rocio (HUVR)

Seville, Spain

Valencia Oncology Institute (IVO)

Valencia, Spain

University and Polytechnic Hospital La Fe

Valencia, Spain

Royal United Hospital, Department of Oncology/Hematology

Bath, United Kingdom

Leicester Royal Infirmary

Leicester, United Kingdom

Royal Marsden Hospital - London

London, United Kingdom

Imperial College Healthcare NHS Trust

London, United Kingdom

The Christie NHS Foundation Trust, Department of Medical Oncology

Manchester, United Kingdom

Churchill Hospital

Oxford, United Kingdom

University Hospital Southampton NHS Foundation Trust

Southampton, United Kingdom

Royal Marsden Hospital - Sutton

Sutton, United Kingdom

Musgrove Park Hospital

Taunton, United Kingdom